《药物动力学与药效学杂志》致力于阐明药物动力学和生物制药在理解药物作用、设计、治疗和评价中的重要性。实验和理论文章处理的主题，如药物处置动力学;临床药物动力学;药物反应的时间过程;以及影响代谢产物形成和分布的因素。原为药物动力学和生物药剂学杂志。
Journal of Pharmacokinetics and Pharmacodynamics is devoted to illustrating the importance of pharmacokinetic and biopharmaceutical applications in the understanding of drug action, design, therapy, and evaluation. Experimental and theoretical articles deal with topics such as the kinetics of drug disposition; clinical pharmacokinetics; the time course of pharmacological response; and factors affecting formation and disposition of metabolites. Formerly Journal of Pharmacokinetics and Biopharmaceutics.